Prezentatsia_Microsoft_PowerPoint

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Groupmeeting
9. 11. 2016
Chizhova Maria
PhD student, 2d year

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10 examples
Dar’in D.; Bakulina O.; Chizhova M.; Krasavin M.
New Heterocyclic Product Space for the
Castagnoli−Cushman Three-Component Reaction.
Org. Lett. 2015, 17, 3930−3933
24 examples
6 X-rays
* Dar'in, D.; Bakulina, O.;
Nikolskaya, S.; Gluzdikov I.;
Krasavin M.
The rare cis-configured
trisubstituted lactam
products obtained by the
Castagnoli–Cushman
reaction in N,Ndimethylformamide. RSC
Adv., 2016, 6, 49411
Chizhova M.; Bakulina O.; Dar’in D.; Krasavin M. New Dicarboxylic Acid Anhydride for Ambient-Temperature
Castagnoli-Cushman Reactions. Chemistry Select, 2016, 1, 5487 – 5492
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Other substrates in CCR
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4.

in process
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5.

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Grintsevich S.
Chizhova M.
Fischer indole synthesis
*Golubev P.; Bakulina O.; Dar'in D.; Krasavin M. Indoline-Based Constrained Peptidomimetic Motifs Obtained via the Joullie–
Ugi Reaction of Indolenines. Eur. J. Org. Chem 2016, 23, 3969-3976
**Estévez V.; Kloeters L.; Kwietniewska N.; Vicente-García E.; Ruijter E.; Orru R. V. A. Ugi-Type Reactions of Spirocyclic
Indolenines as a Platform for Compound Library Generation. Synlett 2016, 27, A–E
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2 ways of CCR
Our plans
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